SCHEMBL19658404

SCHEMBL19658404

CC(=O)N(C)C1CCN(c2cccc(C(C)C)c2)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.58
HRH3 Q9Y5N1 1/20 0.46
NPY5R Q15761 8/20 0.45
PANK3 Q9H999 1/20 0.43
SETD2 Q9BYW2 1/20 0.41
CCR5 P51681 2/20 0.41
MCHR1 Q99705 1/20 0.41
ACACB O00763 1/20 0.41
ADAM10 O14672 1/20 0.40
ITGB2 P05107 1/20 0.40
ICAM1 P05362 1/20 0.40
ITGAL P20701 1/20 0.40
PIK3CD O00329 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19702028 0.93 NOTUM (0.62) NOTUMHRH3SETD2CCR5MCHR1
SCHEMBL19652215 0.89 NOTUM (0.57) NOTUMHRH3NPY5RPANK3CCR5
SCHEMBL19702022 0.85 NOTUM (0.54) NOTUMHRH3NPY5RCCR5ACACB
SCHEMBL19658405 0.84 PANK3 (0.47) HRH3NPY5RPANK3MCHR1
SCHEMBL19658391 0.83 NPY5R (0.60) NOTUMNPY5RSETD2ACACB
SCHEMBL19702020 0.82 CCR5 (0.58) NOTUMHRH3NPY5RCCR5PIK3CD
SCHEMBL14321771 0.82 NPY5R (0.61) NPY5RSETD2MCHR1PIK3CD
SCHEMBL26816763 0.81 NOTUM (0.71) NOTUMHRH3PANK3ACACBADAM10
SCHEMBL19702023 0.81 NOTUM (0.49) NOTUMHRH3NPY5RCCR5ACACB
SCHEMBL19658738 0.81 NPY5R (0.56) NOTUMNPY5RMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2017-12-14 US disclosed
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2017-12-14 US disclosed
US-20170340604-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2017-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS PIK3R3, JAK2, JAK3 NOTUM 3221/4885HRH3 61/4885NPY5R 500/4885
US-20170340604-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF BRD4, BRDT, BRD3 NOTUM 2215/4885HRH3 131/4885NPY5R 1431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.