SCHEMBL19660223

SCHEMBL19660223

C=C(C)/C(C#N)=C(\C)N1CCc2ccccc2C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.54
ALDH1A1 P00352 3/20 0.49
MAPT P10636 2/20 0.49
TAAR1 Q96RJ0 2/20 0.49
ALOX15 P16050 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2D6 P10635 2/20 0.46
MAOA P21397 2/20 0.46
TMPRSS2 O15393 1/20 0.46
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46
SLC6A2 P23975 1/20 0.46
KMT2A Q03164 3/20 0.45
PHGDH O43175 1/20 0.45
MGLL Q99685 1/20 0.45
MEN1 O00255 1/20 0.45
ACE P12821 2/20 0.45
HRH3 Q9Y5N1 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234233 0.85 NOTUM (0.50) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL5234227 0.85 NOTUM (0.50) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL5234219 0.85 NOTUM (0.50) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL20749828 0.78 NOTUM (0.64) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL8244060 0.77 NOTUM (0.68) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL16281586 0.75 NOTUM (0.70) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL21233478 0.72 MAOA (0.59) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL27388745 0.71 NOTUM (0.54) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL30539318 0.71 NOTUM (1.00) NOTUMALDH1A1MAPTTAAR1ALOX15
SCHEMBL3210469 0.71 NOTUM (1.00) NOTUMALDH1A1MAPTTAAR1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017205193-A1 SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS USEFUL AS GPR120 AGONISTS MERCK SHARP & DOHME CORP. (US) 2017-11-30 WO disclosed