SCHEMBL19664982

SCHEMBL19664982

CS(=O)(=O)Nc1ccc(-n2nc(C(F)(F)F)cc2-c2ccc(-c3ccc(F)cc3)cc2)cc1

nearest known ligand 0.98

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.98
PTGS1 P23219 6/20 0.74
CYP2C9 P11712 1/20 0.60
PDPK1 O15530 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698670 0.99 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346838 0.91 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346891 0.91 PTGS2 (0.91) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346857 0.91 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346849 0.90 PTGS2 (0.98) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346767 0.90 PTGS2 (0.98) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15347197 0.90 PTGS2 (0.98) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346938 0.90 PTGS2 (0.83) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL4617859 0.90 PTGS2 (0.83) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL15346533 0.89 PTGS2 (0.78) PTGS2PTGS1CYP2C9PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3363435-A1 ANTI-STAPHYLOCOCCAL CELECOXIB DERIVATIVES The Ohio State University Research Foundation (US) 2018-08-22 EP disclosed
EP-2635274-B1 ANTI-STAPHYLOCOCCAL CELECOXIB DERIVATIVES UNIV OHIO STATE RES FOUND (US) 2017-12-06 EP disclosed