SCHEMBL1967103

SCHEMBL1967103

CN1CCN(CCOc2ccc(C(=O)N3C=C(C(=O)O)c4[nH]c5ccccc5c4C(C)(C)C3)cc2)CC1

nearest known ligand 0.81

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.81
KCNH2 Q12809 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966827 0.96 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1965630 0.92 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1968461 0.92 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1967324 0.90 NR1H4 (0.81) NR1H4KCNH2
SCHEMBL1242993 0.90 NR1H4 (1.00) NR1H4KCNH2
SCHEMBL4758760 0.89 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1965284 0.88 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1967457 0.88 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1967301 0.86 NR1H4 (0.82) NR1H4KCNH2
SCHEMBL1243669 0.86 NR1H4 (1.00) NR1H4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334681-A1 1,2,3,6-TETRAHYDROAZEPINO[4,5-B]INDOLE-5-CARBOXYLATE NUCLEAR RECEPTOR INHIBITORS Wyeth LLC (US) 2011-06-22 EP disclosed
WO-2010036362-A1 1,2,3,6-TETRAHYDROAZEPINO[4,5-B]INDOLE-5-CARBOXYLATE NUCLEAR RECEPTOR INHIBITORS WYETH (US) 2010-04-01 WO disclosed