SCHEMBL19675231

SCHEMBL19675231

COc1ccc2c(c1)N(C(=O)Nc1ccc(C)cc1)CC2

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.67
RAB9A P51151 6/20 0.67
SMN1; SMN2 Q16637 5/20 0.67
NFKB1 P19838 4/20 0.67
NFKB2 Q00653 4/20 0.67
RELA Q04206 4/20 0.67
MAPT P10636 4/20 0.67
PKM P14618 3/20 0.67
MAOB P27338 1/20 0.67
TP53 P04637 4/20 0.67
ROCK1 Q13464 1/20 0.60
HTR2C P28335 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPK1 P28482 1/20 0.52
POLB P06746 2/20 0.51
NOTUM Q6P988 1/20 0.50
HTR2B P41595 1/20 0.49
HTR2A P28223 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19675184 0.89 NPC1 (0.66) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL15897761 0.89 NPC1 (0.66) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL19675326 0.82 NPC1 (0.57) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL4862236 0.82 MAPT (0.64) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL15882082 0.81 NPC1 (0.56) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL17321521 0.81 ROCK1 (0.81) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL12692444 0.81 RAB9A (1.00) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL28367564 0.80 NPC1 (1.00) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL15897878 0.79 ROCK1 (0.59) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL2208006 0.78 NOTUM (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252050-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed
EP-3252049-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed