SCHEMBL19675899

SCHEMBL19675899

Cc1cnc(Cl)nc1Nc1ccc2ncccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.50
EGFR P00533 4/20 0.49
TGFBR1 P36897 1/20 0.47
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
NPC1 O15118 3/20 0.46
POLB P06746 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALDH1A1 P00352 3/20 0.45
PIK3CA P42336 1/20 0.45
MTOR P42345 1/20 0.45
ERBB2 P04626 1/20 0.45
ERBB4 Q15303 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
RAB9A P51151 2/20 0.44
LMNA P02545 1/20 0.44
NOTUM Q6P988 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28481059 0.86 GRM4 (0.52) GRM4EGFRTGFBR1ABCB1ABCC1
SCHEMBL16012778 0.84 EGFR (0.55) GRM4EGFRTGFBR1ABCB1ABCC1
SCHEMBL655954 0.84 GRM4 (0.50) GRM4EGFRTGFBR1ABCB1ABCC1
SCHEMBL15585196 0.84 GRM4 (0.50) GRM4EGFRTGFBR1ABCB1ABCC1
SCHEMBL2627259 0.80 MAPK8 (0.52) GRM4EGFRNPC1POLBMAPT
SCHEMBL16012092 0.79 PIN1 (0.64) GRM4EGFRABCG2NPC1POLB
SCHEMBL2627260 0.79 SYK (0.57) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL264886 0.77 GRM4 (0.48) GRM4EGFRMEN1KMT2ASYK
SCHEMBL265799 0.77 STK17A (0.53) GRM4EGFRMEN1KMT2ASYK
SCHEMBL30306442 0.77 STK17A (0.53) GRM4EGFRMEN1KMT2ASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2840080-B1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2017-12-06 EP disclosed