SCHEMBL19681369

SCHEMBL19681369

COc1c(Br)c(Cl)cc2c(N3CCN(C(=O)O)CC3)ncnc12

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.44
BACE1 P56817 1/20 0.44
PDGFRB P09619 14/20 0.43
PDGFRA P16234 6/20 0.42
KIT P10721 2/20 0.42
FLT3 P36888 2/20 0.42
KRAS P01116 2/20 0.40
EGFR P00533 1/20 0.40
HMOX2 P30519 1/20 0.40
CRYZ Q08257 1/20 0.40
VAT1 Q99536 1/20 0.40
RTN4 Q9NQC3 1/20 0.40
MTNR1B P49286 1/20 0.40
EIF2AK2 P19525 1/20 0.40
ENPP1 P22413 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637088 0.87 KIT (0.49) ACHEBACE1PDGFRBPDGFRAKIT
SCHEMBL18128513 0.86 HRH4 (0.37) ACHEBACE1PDGFRBPDGFRAKIT
SCHEMBL21839499 0.85 KRAS (0.43) ACHEBACE1PDGFRBKITKRAS
SCHEMBL16637086 0.83 PDGFRB (0.36) ACHEBACE1PDGFRBPDGFRAKIT
SCHEMBL16637106 0.83 KRAS (0.51) ACHEBACE1PDGFRBKITKRAS
SCHEMBL19681376 0.79 KRAS (0.46) PDGFRBPDGFRAKRASEGFRHMOX2
SCHEMBL25180032 0.77 ACHE (0.45) ACHEBACE1PDGFRBPDGFRAKIT
SCHEMBL21839989 0.75 PDGFRB (0.49) ACHEBACE1PDGFRBPDGFRAKIT
SCHEMBL21415570 0.74 KIT (0.52) ACHEBACE1KITKRASEGFR
SCHEMBL26967250 0.74 KIT (0.45) KITKRASEGFRHMOX2CRYZ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9840516-B2 Substituted quinazolines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2017-12-12 US disclosed