SCHEMBL19686528

SCHEMBL19686528

Cc1cc(C)n(-c2nc(NC3CCC(F)(F)CC3)cc(C3=CCCOC3)n2)n1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNN2 Q9H2S1 1/20 0.48
KCNN3 Q9UGI6 1/20 0.48
ADORA2A P29274 14/20 0.39
ADORA1 P30542 9/20 0.39
ALOX15 P16050 1/20 0.35
CYP3A4 P08684 2/20 0.35
IDH1 O75874 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21144303 0.83 ADORA2A (0.43) ADORA2AADORA1CYP3A4
SCHEMBL19686611 0.80 KCNN2 (0.58) KCNN2KCNN3ADORA2AADORA1ALOX15
SCHEMBL19686804 0.80 KCNN3 (0.73) KCNN2KCNN3ALOX15POLB
SCHEMBL19686594 0.80 KCNN2 (0.57) KCNN2KCNN3ADORA2AADORA1ALOX15
SCHEMBL19686815 0.79 ADORA2A (0.61) KCNN2KCNN3ADORA2AADORA1ALOX15
SCHEMBL19686522 0.78 KCNN2 (0.58) KCNN2KCNN3ADORA2AADORA1ALOX15
SCHEMBL21144301 0.78 ADORA2A (0.35) ADORA2AADORA1ALOX15CYP3A4
SCHEMBL19686521 0.77 KCNN3 (0.59) KCNN2KCNN3ALOX15IDH1POLB
SCHEMBL19686627 0.76 KCNN2 (0.48) KCNN2KCNN3ADORA2AADORA1ALOX15
SCHEMBL21143845 0.76 KCNN2 (0.48) KCNN2KCNN3ADORA2AADORA1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240317705-A1 POTASSIUM CHANNEL MODULATORS NOVARTIS AG (CH) 2024-09-26 US disclosed
US-10774064-B2 Potassium channel modulators CADENT THERAPEUTICS, INC. (US) 2020-09-15 US disclosed
US-10774064-B2 Potassium channel modulators CADENT THERAPEUTICS, INC. (US) 2020-09-15 US disclosed
US-20190218200-A1 POTASSIUM CHANNEL MODULATORS NOVARTIS AG (CH) 2019-07-18 US disclosed
US-20190218200-A1 POTASSIUM CHANNEL MODULATORS NOVARTIS AG (CH) 2019-07-18 US disclosed
WO-2017139697-A9 BACTERIA ENGINEERED TO TREAT DISEASES ASSOCIATED WITH HYPERAMMONEMIA SYNLOGIC, INC. (US) 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240317705-A1 POTASSIUM CHANNEL MODULATORS KCNJ11, KCNJ2, KCNJ1 KCNN2 5/4885KCNN3 11/4885ADORA2A 1711/4885
US-10774064-B2 Potassium channel modulators KCNJ11, KCNJ2, KCNJ1 KCNN2 5/4885KCNN3 11/4885ADORA2A 1711/4885
US-20190218200-A1 POTASSIUM CHANNEL MODULATORS KCNJ11, KCNJ2, KCNJ1 KCNN2 5/4885KCNN3 11/4885ADORA2A 1711/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.