SCHEMBL1970757

SCHEMBL1970757

Cc1ccccc1-c1sc(Br)nc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.46
NR1H4 Q96RI1 2/20 0.43
MYC P01106 1/20 0.39
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39
IKBKB O14920 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MCL1 Q07820 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
STAT6 P42226 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PIN1 Q13526 1/20 0.36
PRKDC P78527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL269610 0.86 HPGD (0.47) HPGDNR1H4MYCHCRTR1HCRTR2
SCHEMBL8823046 0.82 SMN1; SMN2 (0.51) HPGDALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL3006440 0.81 NPC1 (0.41) HPGDHCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL1340822 0.81 MAPK14 (0.50) HPGDNR1H4MYCIKBKBALDH1A1
SCHEMBL4068223 0.78 KDM4E (0.51) HPGDALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL27814745 0.77 MCL1 (0.43) HCRTR1HCRTR2ALDH1A1MAPTSMN1; SMN2
SCHEMBL1340229 0.76 PIN1 (0.52) IKBKBMEN1KMT2APIN1
SCHEMBL2547639 0.74 KDM4E (0.47) HPGDALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL1340615 0.74 HCRTR1 (0.41) HPGDMYCHCRTR1HCRTR2SMN1; SMN2
SCHEMBL269670 0.74 KMT2A (0.46) HPGDHCRTR1HCRTR2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed