SCHEMBL1972282

SCHEMBL1972282

Clc1ccc(C[C]2CCN(c3ncnc4[nH]cnc34)CC2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 8/20 0.47
AKT1 P31749 5/20 0.39
AKT3 Q9Y243 1/20 0.39
LMNA P02545 1/20 0.39
HTR6 P50406 1/20 0.37
LRRK2 Q5S007 2/20 0.37
GSK3B P49841 3/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CSF1R P07333 1/20 0.35
RECQL P46063 1/20 0.35
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1972518 0.87 AKT2 (0.46) AKT2AKT1AKT3GSK3BCYP2D6
SCHEMBL1972284 0.81 AKT2 (0.48) AKT2LMNAGSK3BCYP2D6RPS6KB1
SCHEMBL1003154 0.80 AKT2 (0.72) AKT2AKT1GSK3BCYP2D6CYP2C9
SCHEMBL1002683 0.78 AKT2 (0.58) AKT2AKT1GSK3BCYP2D6CYP2C9
SCHEMBL3917917 0.74 AKT2 (0.87) AKT2AKT1AKT3GSK3BCYP2D6
SCHEMBL1000907 0.73 AKT1 (0.60) AKT2AKT1GSK3B
SCHEMBL3917914 0.73 AKT2 (0.70) AKT2AKT1AKT3GSK3BCYP2D6
SCHEMBL3931922 0.72 AKT2 (0.70) AKT2AKT1AKT3GSK3BCYP2D6
SCHEMBL6755688 0.72 HTT (0.47) AKT2LMNAGSK3BRECQL
SCHEMBL1791997 0.70 RECQL (0.66) AKT2LMNALRRK2RPS6KB1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812004-B1 ORTHO- CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E. G. PURINES) AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2011-06-22 EP claimed