SCHEMBL19732415

SCHEMBL19732415

COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(=O)CO)C[C@@H]3OC1C[C@H](C)[C@H](O)[C@H](C)O1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.87
KMT2A Q03164 8/20 0.87
THRB P10828 7/20 0.87
BLM P54132 7/20 0.87
RECQL P46063 6/20 0.87
BRCA1 P38398 6/20 0.87
TOP2A P11388 5/20 0.87
TDP1 Q9NUW8 5/20 0.87
HIF1A Q16665 5/20 0.87
SMN1; SMN2 Q16637 5/20 0.87
MAPT P10636 4/20 0.87
MAPK1 P28482 4/20 0.87
CHRM1 P11229 3/20 0.87
TBXA2R P21731 3/20 0.87
KDM4E B2RXH2 3/20 0.87
ALDH1A1 P00352 3/20 0.87
ABCB1 P08183 3/20 0.87
PTGS1 P23219 3/20 0.87
STAT6 P42226 3/20 0.87
HTT P42858 3/20 0.87

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13417668 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL14497179 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL10182791 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL17991858 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL18751202 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL20382875 1.00 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
Hydroxyrubicin SCHEMBL30052370 0.94 MEN1 (0.87) MEN1KMT2ATHRBBLMRECQL
SCHEMBL14497184 0.94 MEN1 (0.77) MEN1KMT2ATHRBBLMRECQL
SCHEMBL3036863 0.94 S100A4 (0.86) MEN1KMT2ATHRBBLMRECQL
SCHEMBL18558770 0.94 MEN1 (0.85) MEN1KMT2ATHRBBLMRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216791-A1 ANTICANCER DRUG CONJUGATES Ariel Scientific Innovations Ltd. (IL) 2017-12-21 WO disclosed