SCHEMBL19734532

SCHEMBL19734532

CC(c1cc(F)cc(F)c1)C1CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
GPR119 Q8TDV5 5/20 0.41
USP30 Q70CQ3 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NR1H2 P55055 1/20 0.40
RORC P51449 3/20 0.39
BACE1 P56817 2/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19734489 0.86 DPP4 (0.42) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL20164106 0.86 DPP4 (0.42) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL19734488 0.86 DPP4 (0.42) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL18249566 0.86 DPP4 (0.42) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL1529076 0.85 DPP4 (0.41) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL19734728 0.84 DPP4 (0.41) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL23830783 0.81 USP30 (0.48) GPR119USP30NPC1ALDH1A1MAPT
SCHEMBL19726039 0.80 DPP4 (0.43) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL19734715 0.80 DPP4 (0.39) DPP4HDAC1HDAC2GPR119USP30
SCHEMBL23212067 0.79 MAPT (0.48) DPP4GPR119USP30NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216280-A1 TETRAHYDRO-PYRIDO[3,4-b]INDOLE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-12-21 WO disclosed