SCHEMBL19734728

SCHEMBL19734728

COC(c1cc(F)cc(F)c1)C1CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
USP30 Q70CQ3 2/20 0.39
PDE4B Q07343 1/20 0.38
NR1H2 P55055 1/20 0.38
GPR119 Q8TDV5 2/20 0.37
RORC P51449 1/20 0.37
MMP13 P45452 1/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.36
THRB P10828 1/20 0.36
NAMPT P43490 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19713486 0.85 DPP4 (0.40) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL19713432 0.84 DPP4 (0.40) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL19734489 0.84 DPP4 (0.42) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL20164106 0.84 DPP4 (0.42) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL18249566 0.84 DPP4 (0.42) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL19734532 0.84 DPP4 (0.42) DPP4HDAC1HDAC2USP30NR1H2
SCHEMBL19734488 0.84 DPP4 (0.42) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL1529076 0.83 DPP4 (0.41) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL19713440 0.81 DPP4 (0.41) DPP4HDAC1HDAC2USP30PDE4B
SCHEMBL15804381 0.79 SLC6A2 (0.52) PDE4BMAPTNPC1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216280-A1 TETRAHYDRO-PYRIDO[3,4-b]INDOLE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-12-21 WO disclosed