SCHEMBL19734593

SCHEMBL19734593

Cc1nc(Cl)c(C#N)c(-c2ccco2)c1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
HSD17B10 Q99714 7/20 0.52
KDM4E B2RXH2 7/20 0.52
POLB P06746 1/20 0.52
HPGD P15428 6/20 0.51
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
CASP1 P29466 1/20 0.51
BLM P54132 1/20 0.51
LMNA P02545 1/20 0.51
MAPT P10636 4/20 0.48
ADORA1 P30542 10/20 0.48
ADORA2A P29274 6/20 0.48
ADORA3 P0DMS8 3/20 0.48
NPSR1 Q6W5P4 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TSHR P16473 1/20 0.46
ADORA2B P29275 2/20 0.46
ALOX15 P16050 2/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19716807 0.89 ADORA1 (0.53) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL23162717 0.77 ADORA2A (0.53) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL29623216 0.77 ADORA2A (0.53) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL21116577 0.73 ALDH1A1 (0.51) ALDH1A1HSD17B10KDM4EPOLBHPGD
Ammonia Solution, Strong SCHEMBL19717396 0.72 ADORA1 (0.50) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL6256113 0.71 HSD17B10 (0.72) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL6258393 0.71 ADORA1 (0.61) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL6440893 0.71 ADORA2A (0.68) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL22889894 0.70 ALDH1A1 (0.46) ALDH1A1HSD17B10KDM4EPOLBHPGD
SCHEMBL6441030 0.70 KDM4E (0.75) ALDH1A1HSD17B10KDM4EPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed