SCHEMBL19734741

SCHEMBL19734741

N#Cc1c(O)nc(ON)c(C#N)c1-c1ccco1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 10/20 0.55
KDM4E B2RXH2 8/20 0.46
ALDH1A1 P00352 8/20 0.46
MEN1 O00255 7/20 0.46
KMT2A Q03164 7/20 0.46
HSD17B10 Q99714 6/20 0.46
HPGD P15428 6/20 0.46
MAPT P10636 4/20 0.46
GAA P10253 2/20 0.46
ALOX15 P16050 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
ADORA2A P29274 6/20 0.45
ADORA3 P0DMS8 3/20 0.45
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 2/20 0.44
RXFP1 Q9HBX9 2/20 0.44
POLB P06746 1/20 0.43
ADORA2B P29275 3/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21116577 0.85 ALDH1A1 (0.51) ADORA1KDM4EALDH1A1MEN1KMT2A
Ammonia Solution, Strong SCHEMBL19717396 0.84 ADORA1 (0.50) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL28737280 0.74 ADORA1 (0.53) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL29658805 0.70 ALDH1A1 (0.46) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL19716807 0.70 ADORA1 (0.53) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL6442269 0.70 ADORA1 (0.74) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL6442224 0.69 ADORA1 (0.59) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL6258393 0.68 ADORA1 (0.61) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL6441455 0.65 ADORA1 (0.66) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL6441030 0.65 KDM4E (0.75) ADORA1KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed