SCHEMBL1973565

SCHEMBL1973565

CC(C)OC1(C(=O)c2ccc3[nH]ncc3c2)CCCN1C

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.52
SLC6A2 P23975 4/20 0.52
SLC6A4 P31645 4/20 0.52
SLC6A3 Q01959 4/20 0.52
ACACB O00763 6/20 0.42
ACACA Q13085 6/20 0.42
KCNH2 Q12809 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CTNNB1 P35222 3/20 0.41
WNT3A P56704 3/20 0.41
CYP3A4 P08684 2/20 0.41
ROCK2 O75116 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
DDR1 Q08345 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442649 0.73 CYP2D6 (0.47) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL414020 0.72 SLC6A2 (0.76) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL31581088 0.70 ACACB (0.48) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL445754 0.70 CYP2D6 (0.55) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL5418713 0.69 ROCK2 (0.58) CYP2D6SLC6A2SLC6A4SLC6A3NPC1
SCHEMBL25139625 0.69 CTNNB1 (0.58) CYP2D6SLC6A2SLC6A4SLC6A3NPC1
SCHEMBL413631 0.68 SLC6A2 (1.00) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL415206 0.68 SLC6A2 (1.00) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL415289 0.68 SLC6A2 (1.00) CYP2D6SLC6A2SLC6A4SLC6A3ACACB
SCHEMBL31581176 0.67 HPGD (0.66) ACACBACACAKCNH2CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102157-B1 HETEROARYL PYRROLIDINYL AND PIPERIDINYL KETONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-06-22 EP claimed