SCHEMBL19737563

SCHEMBL19737563

O=Cc1ccc2nc(-c3cccnc3)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.49
KCNH2 Q12809 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
ERN1 O75460 3/20 0.44
CYP19A1 P11511 2/20 0.44
CYP2A6 P11509 5/20 0.43
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
CYP3A4 P08684 5/20 0.41
CYP2E1 P05181 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2B6 P20813 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP17A1 P05093 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16110536 0.83 NPC1 (0.53) KCNH2HRH3ERN1CYP3A4CYP2C9
SCHEMBL18526967 0.81 HPGD (0.52) TTKERN1CYP19A1CYP2A6HSP90AA1
SCHEMBL23016380 0.79 CYP19A1 (0.58) KCNH2HRH3CYP19A1CYP2A6CYP3A4
SCHEMBL16829469 0.79 ESR1 (0.63) KCNH2HRH3CYP19A1CYP2A6HSP90AA1
SCHEMBL19737512 0.79 CYP2A6 (0.57) KCNH2HRH3CYP19A1CYP2A6CYP3A4
SCHEMBL23016379 0.77 CYP11B2 (0.69) KCNH2HRH3CYP19A1CYP2A6CYP3A4
SCHEMBL31565814 0.76 NPC1 (0.65) CYP19A1CYP2A6HSP90AA1HSP90AB1PTK2
SCHEMBL30804561 0.76 NPC1 (0.65) CYP19A1CYP2A6HSP90AA1HSP90AB1PTK2
SCHEMBL2722439 0.76 NPC1 (0.65) CYP19A1CYP2A6HSP90AA1HSP90AB1PTK2
SCHEMBL23016428 0.76 CYP11B2 (0.58) KCNH2HRH3CYP19A1CYP2A6PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017217439-A1 THIENO[2,3-b]PYRIDINE DERIVATIVE AND QUINOLINE DERIVATIVE, AND USE THEREOF 国立大学法人東京大学 2017-12-21 WO disclosed