SCHEMBL1974487

SCHEMBL1974487

COc1c(N2CCC(OC(=O)O)CC2)c(F)cc2c(=O)c(C(=O)NCc3ccc(Cl)cc3Cl)cn([C@H]3C[C@H]3F)c12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.45
TOP1 P11387 8/20 0.44
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 3/20 0.42
POLB P06746 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HPGD P15428 2/20 0.41
PRKD3 O94806 1/20 0.41
ALOX15 P16050 1/20 0.41
OPRM1 P35372 1/20 0.41
CLK2 P49760 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200702 0.92 KCNH2 (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL12427385 0.92 KCNH2 (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL12427322 0.88 KCNH2 (0.43) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL1974822 0.87 TOP1 (0.48) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL13744891 0.86 KDM4E (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL4257328 0.86 KDM4E (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL966711 0.86 KDM4E (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL12917302 0.86 KDM4E (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL12917329 0.86 KDM4E (0.46) KCNH2TOP1KDM4EALDH1A1POLB
SCHEMBL968143 0.84 EPHX2 (0.40) KCNH2TOP1KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994020-B1 Substituted quinolones III AICURIS GMBH & CO KG (DE) 2011-06-22 EP disclosed