SCHEMBL19746047

SCHEMBL19746047

N#Cc1ccn2cc(Cc3ccccc3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.56
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
KDM4E B2RXH2 6/20 0.41
PKM P14618 1/20 0.40
ALDH1A1 P00352 3/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
BCAT2 O15382 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A3 P47895 1/20 0.38
HSD17B10 Q99714 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12309272 0.80 PDE10A (0.51) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL10066413 0.80 PDE10A (0.54) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL22499333 0.80 PDE10A (0.51) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL1716596 0.78 PDE10A (0.50) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL22775793 0.78 METTL3 (0.46) SMN1; SMN2NPC1RAB9AKDM4EPKM
SCHEMBL5074964 0.78 AKR1B1 (0.49) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL22530925 0.76 PDE10A (0.60) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL14028695 0.76 KDM4E (0.65) PDE10ASMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL7863078 0.75 KDM4E (0.50) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL31423449 0.73 BRD4 (0.47) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222950-A1 3-HETEROCYCLYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO disclosed