SCHEMBL19746690

SCHEMBL19746690

COc1cc(OC)nc(Cn2ccc(-c3noc(C(F)(F)F)n3)cc2=O)n1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 19/20 0.44
HDAC1 Q13547 14/20 0.44
HDAC8 Q9BY41 10/20 0.44
HDAC4 P56524 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19746864 0.87 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19747037 0.85 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19747008 0.84 HDAC6 (0.50) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746010 0.84 HDAC6 (0.49) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746485 0.84 HDAC6 (0.52) HDAC6HDAC1HDAC8
SCHEMBL19746096 0.82 HDAC6 (0.47) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19745956 0.82 HDAC6 (0.45) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746955 0.82 HDAC6 (0.53) HDAC6HDAC1HDAC8
SCHEMBL19746979 0.81 HDAC6 (0.44) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746424 0.80 HDAC6 (0.50) HDAC6HDAC1HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222952-A1 3- HETEROARYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO claimed