SCHEMBL19752467

SCHEMBL19752467

Cc1ccc(-c2ccc(N(c3ccccc3)c3ccc(C4C=CC=CC4)cc3)cc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
APP P05067 1/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPT P10636 2/20 0.31
CYP2C19 P33261 2/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ACHE P22303 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
EGFR P00533 1/20 0.30
ERBB2 P04626 1/20 0.30
ERBB3 P21860 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23544007 0.97 MAOB (0.35) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL23543669 0.96 APP (0.34) APPALDH1A1KDM4EMAPTCYP2C19
SCHEMBL16994133 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL20686440 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL20714278 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL16500713 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL18774190 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL19443921 0.92 ALDH1A1 (0.34) MAOBAPPALDH1A1KDM4EMAPT
SCHEMBL22755852 0.90 KDM1A (0.35) MAOBALDH1A1KDM4EMAPTCYP2C19
SCHEMBL14067605 0.90 KDM1A (0.35) MAOBALDH1A1KDM4EMAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3260438-A1 DOUBLE-SPIRO TYPE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CONTAINING SAME LG Chem, Ltd. (KR) 2017-12-27 EP disclosed