SCHEMBL1975320

SCHEMBL1975320

O=C(c1cc2cccc(F)c2s1)C1(CC2CCOCC2)CCNC1.O=C(c1cc2cccc(F)c2s1)C1(CC2CCOCC2)CCNC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.44
SLC6A4 P31645 12/20 0.44
SLC6A3 Q01959 12/20 0.44
CYP2D6 P10635 11/20 0.44
CHRNA7 P36544 7/20 0.41
HTR3A P46098 2/20 0.41
CHRNA1 P02708 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA4 P43681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL414018 1.00 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL415193 0.87 CYP2D6 (0.46) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL415153 0.84 CYP2D6 (0.62) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL17707481 0.81 CHRNA7 (0.43) CHRNA7HTR3A
SCHEMBL413703 0.80 CYP2D6 (0.56) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL414183 0.79 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL414182 0.79 CYP2D6 (0.55) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL415192 0.79 CYP2D6 (0.71) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL15423304 0.78 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3CYP2D6CHRNA7
SCHEMBL413109 0.77 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102157-B1 HETEROARYL PYRROLIDINYL AND PIPERIDINYL KETONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-06-22 EP disclosed