SCHEMBL17707481

SCHEMBL17707481

O=C(O)N1CCC(CC2CCOCC2)(C(=O)c2cc3cccc(F)c3s2)C1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 15/20 0.43
HTR3A P46098 10/20 0.43
RORC P51449 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415417 0.88 CHRNA7 (0.39) CHRNA7HTR3ARORCMEN1KMT2A
SCHEMBL1975320 0.81 SLC6A2 (0.44) CHRNA7HTR3A
SCHEMBL414018 0.81 SLC6A2 (0.44) CHRNA7HTR3A
SCHEMBL15423390 0.80 CHRNA7 (0.38) CHRNA7HTR3ARORCMEN1KMT2A
SCHEMBL1971670 0.79 CHRNA7 (0.36) CHRNA7HTR3ARORCHTT
SCHEMBL15423391 0.68 GPR119 (0.37) CHRNA7HTR3ARORC
SCHEMBL415193 0.67 CYP2D6 (0.46) CHRNA7L3MBTL1POLB
SCHEMBL415153 0.65 CYP2D6 (0.62) CHRNA7HTR3AL3MBTL1
SCHEMBL12350297 0.64 CHRNA7 (0.42) CHRNA7HTR3AL3MBTL1
SCHEMBL2889881 0.63 BCL2L1 (0.53) CHRNA7HTR3AL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed