SCHEMBL19775232

SCHEMBL19775232

CCOC(=O)c1ccc(C(=O)CC(O)C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAOA P21397 1/20 0.50
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
PDK3 Q15120 1/20 0.47
PDK4 Q16654 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6902380 0.82 GSK3B (0.48) CA2LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL6902376 0.82 GSK3B (0.48) CA2LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL11900204 0.79 CA1 (0.59) CA12CA1CA2CA7CA9
SCHEMBL6900403 0.78 HDAC3 (0.53) LMNAALDH1A1HTTNPC1MAPT
SCHEMBL6900410 0.78 HDAC3 (0.53) LMNAALDH1A1HTTNPC1MAPT
SCHEMBL27647572 0.78 CA1 (0.79) CA12CA1CA2CA7CA9
SCHEMBL87450 0.76 CA1 (0.83) CA12CA1CA2CA7CA9
SCHEMBL6904340 0.76 GSK3B (0.50) LMNAKMT2AALDH1A1NPC1MAPT
SCHEMBL6900441 0.76 GSK3B (0.50) LMNAKMT2AALDH1A1NPC1MAPT
SCHEMBL6897949 0.75 TSHR (0.55) LMNACYP1A2CYP3A4KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2182809-B1 THERAPEUTIC ISOXAZOLE COMPOUNDS DART NEUROSCIENCE (CAYMAN) LTD (KY) 2018-01-17 EP disclosed