SCHEMBL19781506

SCHEMBL19781506

CC(=O)c1ccc(-c2cc3c(cn2)ncn3-c2ccc(OC(C)C)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 4/20 0.49
KCNH2 Q12809 2/20 0.48
GSK3B P49841 1/20 0.43
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.41
PIM3 Q86V86 2/20 0.41
RAB9A P51151 1/20 0.40
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MCL1 Q07820 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19781537 0.90 KCNH2 (0.55) FGFR1KCNH2GSK3BALDH1A1HPGD
SCHEMBL19781512 0.86 FGFR1 (0.52) FGFR1GSK3BALDH1A1HPGD
SCHEMBL19781604 0.83 KCNH2 (0.48) FGFR1KCNH2ALDH1A1HPGDMAPT
SCHEMBL21449908 0.80 DYRK1A (0.55) FGFR1PIM3RAB9AMAPTKMT2A
SCHEMBL21449942 0.78 GABRP (0.49) FGFR1KCNH2ALDH1A1MAPT
SCHEMBL29636286 0.75 FGFR1 (0.56) FGFR1KCNH2GSK3BALDH1A1HPGD
SCHEMBL19781595 0.75 FGFR1 (0.56) FGFR1KCNH2GSK3BALDH1A1HPGD
SCHEMBL19781511 0.75 FGFR1 (0.59) FGFR1GSK3BALDH1A1HPGDMAPT
SCHEMBL23535517 0.74 FGFR1 (0.61) FGFR1HPGDMAPTKMT2A
SCHEMBL30014068 0.74 FGFR1 (0.61) FGFR1HPGDMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352328-B2 Heterocyclic compounds for the treatment of arenavirus ARISAN THERAPEUTICS INC. (US) 2022-06-07 US disclosed
US-20190308938-A1 Heterocyclic Compounds for the Treatment of Arenavirus NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-10-10 US disclosed
WO-2018013430-A2 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS INC. (US) 2018-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11352328-B2 Heterocyclic compounds for the treatment of arenavirus C9, C1R, C1S FGFR1 3928/4885KCNH2 107/4885GSK3B 4217/4885
US-20190308938-A1 Heterocyclic Compounds for the Treatment of Arenavirus C9, C1R, C1S FGFR1 3928/4885KCNH2 107/4885GSK3B 4217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.