SCHEMBL19781690

SCHEMBL19781690

COC(=N)C(C#N)CC(=O)OC

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.32
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1752393 0.80 TSHR (0.37) TSHRHTTHSD17B10MGAMGAA
SCHEMBL28289211 0.78 TSHR (0.36) TSHRHTTHSD17B10MGAMGAA
SCHEMBL22113432 0.73 TSHR (0.42) TSHRHTTHSD17B10MGAMGAA
SCHEMBL20382939 0.71
SCHEMBL19233797 0.71 TSHR (0.40) TSHRHTTHSD17B10MGAMGAA
SCHEMBL22649369 0.69 TSHR (0.39) TSHRHSD17B10MGAMGAASI
SCHEMBL27392936 0.68 TSHR (0.37) TSHRHTTHSD17B10MGAMGAA
SCHEMBL23175627 0.68 GAA (0.45) TSHRHSD17B10MGAMGAASI
SCHEMBL5077875 0.67 TSHR (0.50) TSHRHTTHSD17B10MGAMGAA
SCHEMBL5081302 0.67 TSHR (0.50) TSHRHTTHSD17B10MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018011160-A1 6,7-DIHYDRO-4H-PYRAZOLO[1,5-A]PYRAZINE COMPOUNDS FOR THE TREATMENT OF INFECTIOUS DISEASES F. HOFFMANN-LA ROCHE AG (CH) 2018-01-18 WO disclosed