SCHEMBL1978206

SCHEMBL1978206

COc1ccc2[nH]c3cnc(-c4cnn(C)c4)cc3c2c1-c1ccc(C(=O)NC2CCCC2N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARK3 P27448 4/20 0.40
CDK2 P24941 2/20 0.39
CCNA2 P20248 1/20 0.39
TTK P33981 1/20 0.39
AXL P30530 9/20 0.39
MERTK Q12866 9/20 0.39
GSK3B P49841 2/20 0.39
DYRK1A Q13627 2/20 0.39
JAK2 O60674 2/20 0.38
SGK1 O00141 1/20 0.38
PIK3CD O00329 1/20 0.38
CHEK1 O14757 1/20 0.38
MAPK13 O15264 1/20 0.38
PDPK1 O15530 1/20 0.38
NUAK1 O60285 1/20 0.38
CCNT1 O60563 1/20 0.38
ROCK2 O75116 1/20 0.38
CHEK2 O96017 1/20 0.38
ABL1 P00519 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12597221 0.99 GSK3B (0.40) MARK3CDK2CCNA2TTKAXL
SCHEMBL12597806 0.93 GSK3B (0.39) MARK3CDK2AXLMERTKGSK3B
SCHEMBL12597407 0.92 GSK3B (0.39) MARK3CDK2AXLMERTKGSK3B
SCHEMBL11908405 0.91 MARK3 (0.40) MARK3CDK2CCNA2TTKAXL
SCHEMBL11907769 0.86 MERTK (0.39) MARK3CDK2AXLMERTKGSK3B
SCHEMBL12597423 0.84 PIM1 (0.43) MARK3CDK2AXLMERTKGSK3B
SCHEMBL3723670 0.83 CHRM1 (0.42) MARK3CDK2AXLMERTKGSK3B
SCHEMBL11929500 0.83 CHRM1 (0.42) MARK3CDK2AXLMERTKGSK3B
SCHEMBL1982173 0.83 CHEK1 (0.45) CDK2CCNA2TTKCHEK1NTRK1
SCHEMBL11909077 0.83 MARK3 (0.43) MARK3CDK2AXLMERTKGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed