SCHEMBL19782773

SCHEMBL19782773

Cc1cc(Br)c2ncc(CCc3ccccc3)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
NOS3 P29474 1/20 0.38
MAPT P10636 1/20 0.36
MAOB P27338 1/20 0.36
CCR1 P32246 2/20 0.36
CCR5 P51681 2/20 0.36
CCR8 P51685 2/20 0.36
ATP4A P20648 1/20 0.35
ATP4B P51164 1/20 0.35
KCNH2 Q12809 1/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PLAU P00749 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23552159 0.84 KCNH2 (0.36) KCNH2NPC1TDP1PLAUKDM4E
SCHEMBL19776515 0.79 PDGFRB (0.50) MAPTMAOBRAB9ANPC1L3MBTL1
SCHEMBL29481808 0.79 PDGFRB (0.50) MAPTMAOBRAB9ANPC1L3MBTL1
SCHEMBL19783279 0.78 CCR1 (0.36) CCR1CCR5CCR8KDM4EHPGD
SCHEMBL30189953 0.76 CCR1 (0.34) MAPTCCR1CCR5CCR8ALDH1A1
SCHEMBL19782862 0.76 CCR1 (0.34) MAPTCCR1CCR5CCR8ALDH1A1
SCHEMBL19783610 0.70 TLR7 (0.32) CCR1CCR5CCR8
SCHEMBL13045274 0.70 KCNH2 (0.47) MAOBKCNH2TDP1PLAUALDH1A1
SCHEMBL19776262 0.69 PRNP (0.40) MAPTCCR1CCR5CCR8RAB9A
SCHEMBL19783078 0.68 CYP11B1 (0.35) MAPTCCR1CCR5CCR8TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed