SCHEMBL19783101

SCHEMBL19783101

CC(C)(C)OC(=O)NCCOc1cc(C(F)(F)F)c2nc(Br)sc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.43
CA1 P00915 5/20 0.43
CA2 P00918 5/20 0.43
CA9 Q16790 5/20 0.43
PDK2 Q15119 1/20 0.43
CACNA1H O95180 1/20 0.42
CACNA1B Q00975 1/20 0.42
CACNA1C Q13936 1/20 0.42
FPR3 P25089 2/20 0.35
FPR2 P25090 2/20 0.35
CFTR P13569 1/20 0.35
SCN9A Q15858 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ITK Q08881 2/20 0.34
EGFR P00533 1/20 0.34
STK17B O94768 1/20 0.34
STK17A Q9UEE5 1/20 0.34
DYRK1A Q13627 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30189817 1.00 CA12 (0.43) CA12CA1CA2CA9PDK2
SCHEMBL19782854 0.89 CA12 (0.44) CA12CA1CA2CA9PDK2
SCHEMBL30189719 0.89 CA12 (0.44) CA12CA1CA2CA9PDK2
SCHEMBL19782843 0.88 CA12 (0.44) CA12CA1CA2CA9PDK2
SCHEMBL21395510 0.86 CA12 (0.45) CA12CA1CA2CA9PDK2
SCHEMBL30189776 0.86 CA12 (0.45) CA12CA1CA2CA9PDK2
SCHEMBL21379504 0.86 CFTR (0.36) CACNA1BCFTRSCN9A
SCHEMBL19782885 0.85 CA12 (0.44) CA12CA1CA2CA9PDK2
SCHEMBL30189608 0.85 CA12 (0.44) CA12CA1CA2CA9PDK2
SCHEMBL19783253 0.82 CA12 (0.41) CA12CA1CA2CA9PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed