SCHEMBL19783253

SCHEMBL19783253

CC(C)(C)OC(=O)NCCOc1cc(C2CC2)c2nc(Br)sc2c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.41
CA1 P00915 5/20 0.41
CA2 P00918 5/20 0.41
CA9 Q16790 5/20 0.41
FPR3 P25089 2/20 0.40
FPR2 P25090 2/20 0.40
PDK2 Q15119 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
SIRT3 Q9NTG7 1/20 0.36
SYK P43405 1/20 0.35
F2R P25116 1/20 0.35
IGF1R P08069 1/20 0.34
SLC5A1 P13866 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
PBK Q96KB5 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30189776 0.85 CA12 (0.45) CA12CA1CA2CA9FPR3
SCHEMBL21395510 0.85 CA12 (0.45) CA12CA1CA2CA9FPR3
SCHEMBL19782843 0.84 CA12 (0.44) CA12CA1CA2CA9FPR3
SCHEMBL19782885 0.84 CA12 (0.44) CA12CA1CA2CA9FPR3
SCHEMBL30189608 0.84 CA12 (0.44) CA12CA1CA2CA9FPR3
SCHEMBL30189817 0.82 CA12 (0.43) CA12CA1CA2CA9FPR3
SCHEMBL19783101 0.82 CA12 (0.43) CA12CA1CA2CA9FPR3
SCHEMBL30189530 0.78 F2RL3 (0.54)
SCHEMBL19783094 0.78 F2RL3 (0.54)
SCHEMBL19783453 0.76 SCN9A (0.41) CA12CA1CA2CA9FPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed