SCHEMBL19783491

SCHEMBL19783491

CCNC(=O)c1cn(-c2ncc(F)cc2F)c2nc(Cl)ccc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.39
CSF1R P07333 2/20 0.38
MEN1 O00255 3/20 0.36
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 1/20 0.36
MAPK8 P45983 1/20 0.36
LMNA P02545 2/20 0.35
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35
NFKB1 P19838 1/20 0.35
HTT P42858 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
PDE4A P27815 1/20 0.35
KCNH2 Q12809 1/20 0.35
EPHA2 P29317 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22590976 0.87 KDM4E (0.39) ALDH1A1HSD17B10TSHRLMNAKDM4E
SCHEMBL19784020 0.85 PDE4A (0.37) ALDH1A1HSD17B10MAPK8LMNAKDM4E
SCHEMBL19784013 0.85 GSK3B (0.35) KMT2AMEN1ALDH1A1HSD17B10MAPK8
SCHEMBL20969353 0.85 GSK3B (0.35) KMT2AMEN1ALDH1A1HSD17B10MAPK8
SCHEMBL19784014 0.85 GSK3B (0.35) KMT2AMEN1ALDH1A1HSD17B10MAPK8
SCHEMBL19784152 0.85 EPHA2 (0.46) KMT2AMEN1ALDH1A1HSD17B10LMNA
SCHEMBL19783901 0.85 EPHA2 (0.38) KMT2AALDH1A1HSD17B10MAPK8LMNA
SCHEMBL19784012 0.85 MAPT (0.43) KMT2ACSF1RMEN1ALDH1A1TSHR
SCHEMBL19784177 0.84 LMNA (0.34) KMT2AMEN1ALDH1A1HSD17B10MAPK8
SCHEMBL20969339 0.84 KMT2A (0.33) KMT2AMEN1ALDH1A1HSD17B10MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018011017-A1 7-SUBSTITUTED 1-PYRIDYL-NAPHTHYRIDINE-3-CARBOXYLIC ACID AMIDES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-01-18 WO disclosed