SCHEMBL19783682

SCHEMBL19783682

COc1cc(C(C)=O)c(N)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 3/20 0.51
SIRT6 Q8N6T7 1/20 0.43
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.38
PABPC1 P11940 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MTNR1A P48039 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31663020 1.00 NNMT (0.51) NNMTSIRT6PIK3CAMTORMKNK1
SCHEMBL17888603 0.86 NNMT (0.56) NNMTSIRT6PIK3CAMTORMKNK1
SCHEMBL29589415 0.86 NNMT (0.51) NNMTSIRT6MKNK1MKNK2MEN1
SCHEMBL2002960 0.86 NNMT (0.51) NNMTSIRT6MKNK1MKNK2MEN1
SCHEMBL31693169 0.86 NNMT (0.65) NNMTSIRT6MKNK1MKNK2MEN1
SCHEMBL15359911 0.84 KDM4E (0.54) NNMTSIRT6MEN1KMT2AKDM4E
SCHEMBL31582715 0.84 KDM4E (0.54) NNMTSIRT6MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL20771312 0.83 KDM4E (0.53) NNMTSIRT6MEN1KMT2AKDM4E
SCHEMBL16701908 0.79 NNMT (0.47) NNMTSIRT6MKNK1MKNK2HTT
SCHEMBL25082752 0.78 SMN1; SMN2 (0.36) NNMTHTTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed