SCHEMBL19785451

SCHEMBL19785451

CNc1nccc(Br)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
LRRK2 Q5S007 2/20 0.37
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
CSNK2A1 P68400 1/20 0.35
HIPK2 Q9H2X6 1/20 0.35
PRKCI P41743 1/20 0.34
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DAO P14920 1/20 0.32
NPC1 O15118 2/20 0.32
JAK2 O60674 1/20 0.31
PTPN11 Q06124 1/20 0.30
KCNH2 Q12809 1/20 0.30
PDCD1 Q15116 2/20 0.30
CD274 Q9NZQ7 2/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785099 0.79 KDM4E (0.39) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL28576286 0.78 KDM4E (0.41) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL30897222 0.78 KDM4E (0.38) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL29211872 0.78 KDM4E (0.38) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL29006810 0.77 CSNK2A1 (0.35) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL21921077 0.77 KDM4E (0.40) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL21575418 0.75 CSNK2A1 (0.35) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL22440558 0.75 KDM4E (0.39) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL22440534 0.73 KDM4E (0.38) KDM4EALDH1A1LMNATDP1LRRK2
SCHEMBL31288549 0.73 KDM4E (0.38) KDM4EALDH1A1LMNATDP1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175081-A1 SHP2 INHIBITOR COMPOUND AND USE THEREOF 深圳真实生物医药科技有限公司 2024-08-29 WO disclosed
WO-2018013597-A1 2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS Revolution Medicines, Inc. (US) 2018-01-18 WO disclosed