SCHEMBL1978738

SCHEMBL1978738

O=C1NC(=O)C2(CC(C3CC3)Oc3ccc(Br)cc32)N1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 7/20 0.48
AKR1B10 O60218 2/20 0.48
AKR1A1 P14550 2/20 0.48
MAPT P10636 1/20 0.41
BACE1 P56817 3/20 0.37
APP P05067 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1820001 0.94 AKR1B1 (0.46) AKR1B1AKR1B10AKR1A1MAPTBACE1
SCHEMBL1822217 0.87 BACE1 (0.54) AKR1B1AKR1B10AKR1A1MAPTBACE1
SCHEMBL1822354 0.86 BACE1 (0.55) AKR1B1AKR1B10AKR1A1MAPTBACE1
SCHEMBL1820144 0.83 BACE1 (0.39) AKR1B1AKR1B10AKR1A1BACE1APP
SCHEMBL25892734 0.82 AKR1B1 (0.63) AKR1B1AKR1B10AKR1A1
SCHEMBL25893192 0.80 AKR1B1 (0.75) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL7949195 0.79 AKR1B1 (0.40) AKR1B1AKR1B10AKR1A1
SCHEMBL1822778 0.79 AKR1B1 (0.47) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL1822427 0.77 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL1979448 0.77 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1MAPTBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed