SCHEMBL1979448

SCHEMBL1979448

O=C1NC(=O)C2(CC(Cc3ccccc3)Oc3ccc(Br)cc32)N1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.45
AKR1B10 O60218 2/20 0.45
AKR1A1 P14550 2/20 0.45
BACE1 P56817 2/20 0.40
KCNH2 Q12809 1/20 0.40
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1822778 0.82 AKR1B1 (0.47) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL7958615 0.80 AKR1B1 (0.43) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL25892734 0.79 AKR1B1 (0.63) AKR1B1AKR1B10AKR1A1
SCHEMBL1978738 0.77 AKR1B1 (0.48) AKR1B1AKR1B10AKR1A1BACE1MAPT
SCHEMBL1823883 0.76 AKR1B1 (0.48) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL9181175 0.76 AKR1B1 (0.65) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL25893192 0.76 AKR1B1 (0.75) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10487420 0.74 AKR1B1 (0.66) AKR1B1
SCHEMBL9818912 0.74 AKR1B1 (0.66) AKR1B1
SCHEMBL9818906 0.74 AKR1B1 (0.66) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed