SCHEMBL19789918

SCHEMBL19789918

CC(C)(C)OC(=O)N1CCCC[C@H]1c1ncc(-c2ccc(-c3ccc(-c4cnc([C@@H]5CCCN5C(=O)OC(C)(C)C)[nH]4)cc3)cc2)[nH]1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.58
CYP2C9 P11712 3/20 0.58
KCNH2 Q12809 2/20 0.58
NR1I2 O75469 1/20 0.58
ABCB11 O95342 1/20 0.58
OPRK1 P41145 1/20 0.58
PRCP P42785 7/20 0.56
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 1/20 0.54
HPGDS O60760 3/20 0.52
OPRM1 P35372 1/20 0.48
OPRD1 P41143 1/20 0.48
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11910995 0.98 CYP3A4 (0.60) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL753302 0.98 CYP3A4 (0.60) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL2706110 0.97 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL10177193 0.95 HPGDS (0.57) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL725968 0.94 PRCP (0.64) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL10145019 0.94 PRCP (0.64) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL23247528 0.94 PRCP (0.57) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL29666028 0.94 PRCP (0.57) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL203852 0.94 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL20401814 0.94 CYP3A4 (0.56) CYP3A4CYP2C9KCNH2NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042901-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB HOLDINGS IRELAND (CH) 2018-01-24 EP disclosed