SCHEMBL1979050

SCHEMBL1979050

C[C@@H]1CC2(NC(=S)NC2=O)c2cc(Br)ccc2O1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 13/20 0.49
PBRM1 Q86U86 1/20 0.42
AKR1B10 O60218 1/20 0.38
AKR1A1 P14550 1/20 0.38
BACE1 P56817 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25892734 0.88 AKR1B1 (0.63) AKR1B1PBRM1AKR1B10AKR1A1
SCHEMBL1821671 0.81 ALOX12 (0.39) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL1820144 0.81 BACE1 (0.39) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL1824927 0.80 AKR1B1 (0.37) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL1824168 0.80 AKR1B1 (0.43) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL7957154 0.80 SIRT2 (0.35) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL1825508 0.78 MAPT (0.34) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL1820450 0.78 AKR1B1 (0.38) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL2377131 0.78 BACE1 (0.54) AKR1B1AKR1B10AKR1A1BACE1
SCHEMBL7948443 0.78 BACE1 (0.37) AKR1B1PBRM1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed