SCHEMBL19791889

SCHEMBL19791889

O=C=Nc1cc2c(c3c1CCCC3)CCC2

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.35
TRPA1 O75762 1/20 0.35
NLRP3 Q96P20 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30120778 0.98 CYP3A4 (0.36) CYP3A4TRPA1ALDH1A1HPGDTDP1
SCHEMBL19791885 0.98 CYP3A4 (0.36) CYP3A4TRPA1ALDH1A1HPGDTDP1
SCHEMBL11103476 0.79 CYP3A4 (0.46) CYP3A4TRPA1TDP1
SCHEMBL19791962 0.78 TRPA1 (0.32) CYP3A4TRPA1NLRP3ALDH1A1
SCHEMBL22012689 0.78 PARP1 (0.32) CYP3A4TRPA1
SCHEMBL19791887 0.76 TRPA1 (0.30) CYP3A4TRPA1
SCHEMBL6867779 0.76 TRPA1 (0.33) CYP3A4TRPA1NLRP3ALDH1A1
SCHEMBL19791775 0.75 TRPA1 (0.32) CYP3A4TRPA1
SCHEMBL20681025 0.74 TRPA1 (0.32) CYP3A4TRPA1NLRP3ALDH1A1
SCHEMBL9709998 0.73 CYP3A4 (0.37) CYP3A4TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018015445-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-25 WO disclosed
EP-3272739-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-24 EP disclosed
EP-3272739-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-24 EP disclosed