Formic Acid

Formic Acid

SCHEMBL1979645

CCc1ocnc1C(=O)Nc1ccc(F)c([C@@]2(C)OC(N)=NC(C)(C)C2(F)F)c1.O=CO

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.45
BACE2 Q9Y5Z0 8/20 0.45
CYP2D6 P10635 1/20 0.44
CTSD P07339 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL1973659 0.88 BACE1 (0.51) BACE1BACE2CTSD
Formic Acid SCHEMBL1980427 0.87 BACE1 (0.45) BACE1BACE2CYP2D6CTSD
Formic Acid SCHEMBL1978067 0.83 BACE1 (0.67) BACE1BACE2
Formic Acid SCHEMBL1978065 0.83 BACE1 (0.67) BACE1BACE2
SCHEMBL1981020 0.79 BACE1 (0.67) BACE1BACE2CYP2D6
SCHEMBL12587602 0.79 BACE1 (0.71) BACE1BACE2
Hydrochloric Acid SCHEMBL1979781 0.78 BACE1 (0.66) BACE1BACE2CYP2D6
SCHEMBL1980888 0.78 BACE1 (0.66) BACE1BACE2CYP2D6
SCHEMBL1980007 0.77 BACE1 (0.68) BACE1BACE2CYP2D6
SCHEMBL1978880 0.77 BACE1 (0.62) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011069934-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-16 WO disclosed