SCHEMBL19797158

SCHEMBL19797158

CCOC(=O)C1=CC(C)CCC1[S+]([O-])Cc1ccc(F)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 8/20 0.43
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
P2RX7 Q99572 5/20 0.37
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
POLB P06746 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19797160 0.77 TLR4 (0.50) TLR4HTTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL19797157 0.77 TLR4 (0.50) TLR4HTTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL21218154 0.70 TLR4 (0.44) TLR4HTTSMN1; SMN2P2RX7L3MBTL1
SCHEMBL28531536 0.70 TLR4 (0.44) TLR4HTTSMN1; SMN2P2RX7L3MBTL1
SCHEMBL21142094 0.67 TLR4 (0.50) TLR4HTTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL21218153 0.67 TLR4 (0.50) TLR4HTTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL19982519 0.66 TLR4 (0.41) TLR4HTTSMN1; SMN2P2RX7L3MBTL1
SCHEMBL19982521 0.66 TLR4 (0.41) TLR4HTTSMN1; SMN2P2RX7L3MBTL1
SCHEMBL872462 0.66 TLR4 (0.56) TLR4HTTSMN1; SMN2P2RX7L3MBTL1
SCHEMBL19982402 0.66 TLR4 (0.36) TLR4HTTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018016657-A1 ETHYL 6-[(2-CHLORO-4-FLUOROPHENYL)METHANESULFONYL]-3-METHYLCYCLOHEX-1-ENE-1-CARBOXYLATE AS TLR4 ANTAGONIST TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-01-25 WO disclosed