SCHEMBL19823046

SCHEMBL19823046

CSC1CN(Cc2ccc(-c3cccn4nc(NC(=O)C5CC5)nc34)cc2)C1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 17/20 0.77
JAK2 O60674 7/20 0.51
JAK3 P52333 4/20 0.49
PTK2 Q05397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24062654 0.90 JAK1 (0.80) JAK1JAK2JAK3PTK2
SCHEMBL19823050 0.87 JAK1 (1.00) JAK1JAK2JAK3PTK2
SCHEMBL19823061 0.86 JAK1 (0.75) JAK1JAK2JAK3
SCHEMBL21044824 0.86 JAK1 (1.00) JAK1JAK2JAK3PTK2
SCHEMBL19823062 0.85 JAK1 (0.75) JAK1JAK2JAK3PTK2
SCHEMBL13535559 0.85 JAK1 (0.73) JAK1JAK2JAK3PTK2
SCHEMBL21044823 0.85 JAK1 (0.84) JAK1JAK2JAK3PTK2
SCHEMBL24062649 0.84 JAK1 (0.72) JAK1JAK2JAK3
SCHEMBL13535409 0.82 JAK1 (0.70) JAK1JAK2
SCHEMBL13535386 0.81 JAK1 (0.72) JAK1JAK2JAK3PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018019223-A1 COMPOUND AS SELECTIVE JAK INHIBITOR, AND SALT AND THERAPEUTIC USE THEREOF 张文燕 2018-02-01 WO disclosed