SCHEMBL19852570

SCHEMBL19852570

CCCC1(C)C=Cc2cnccc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.40
PTGS2 P35354 1/20 0.40
XDH P47989 1/20 0.40
TRPA1 O75762 1/20 0.33
LDHA P00338 1/20 0.33
CNR1 P21554 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CNR2 P34972 1/20 0.33
SLC6A3 Q01959 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
TRPV2 Q9Y5S1 1/20 0.33
BACE1 P56817 1/20 0.32
ALOX5 P09917 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2E1 P05181 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810009 0.77 HIF1A (0.41) PTGS1PTGS2XDHCYP3A4
SCHEMBL4799682 0.73 PTGS1 (0.50) PTGS1PTGS2XDHTRPA1LDHA
SCHEMBL4795100 0.67 PTGS1 (0.40) PTGS1PTGS2XDHTRPA1LDHA
SCHEMBL30236360 0.65
SCHEMBL14178670 0.65 HIF1A (0.47) PTGS1PTGS2XDHBACE1
SCHEMBL1078099 0.64 SLC6A2 (0.38) PTGS1PTGS2XDHTRPA1LDHA
SCHEMBL14178667 0.64 HIF1A (0.48) PTGS1PTGS2XDH
SCHEMBL7300006 0.64 HIF1A (0.41) CYP3A4
SCHEMBL2558890 0.64 PTGS1 (0.46) PTGS1PTGS2XDHBACE1
SCHEMBL8910299 0.64 CYP17A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed