SCHEMBL19853062

SCHEMBL19853062

CCCCCCCC(CCCC)c1ncc(F)cn1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DNM1 Q05193 2/20 0.34
NR1I2 O75469 1/20 0.33
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.31
SLC2A1 P11166 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23869504 0.98 NR1I2 (0.34) DNM1NR1I2MAPTLMNASLC2A1
SCHEMBL21346764 0.98 NR1I2 (0.34) DNM1NR1I2MAPTLMNASLC2A1
SCHEMBL19965631 0.87 NR1I2 (0.31) NR1I2
SCHEMBL27100721 0.82 DNM1 (0.34) DNM1NR1I2LMNASLC2A1CA2
SCHEMBL19231984 0.82 DNM1 (0.34) DNM1NR1I2MAPTLMNASLC2A1
SCHEMBL22810433 0.81
SCHEMBL24805811 0.80 DEGS1 (0.39) NR1I2MAPTLMNA
SCHEMBL19987514 0.80 NR1I2 (0.34) DNM1NR1I2MAPTLMNASLC2A1
SCHEMBL19134116 0.79 DNM1 (0.38) DNM1NR1I2LMNA
SCHEMBL21725999 0.79 POLB (0.33) NR1I2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10196399-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof SUNOVION PHARMACEUTICALS INC. (US) 2019-02-05 US disclosed
US-20180037585-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF SUNOVION PHARAMCEUTICALS INC. 2018-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10196399-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof GRM5, GRIK5, GRM2 DNM1 732/4885NR1I2 723/4885MAPT 4094/4885
US-20180037585-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF GRM5, GRIK5, GRM2 DNM1 732/4885NR1I2 723/4885MAPT 4094/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.