SCHEMBL19860068

SCHEMBL19860068

CC(C)c1ccc(C(=O)Nc2cccc(Oc3ccccc3)c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.64
HPSE Q9Y251 1/20 0.61
RAB9A P51151 6/20 0.60
NPC1 O15118 5/20 0.60
NLRP3 Q96P20 1/20 0.60
PLAU P00749 1/20 0.59
TRPV1 Q8NER1 1/20 0.59
GALK1 P51570 1/20 0.58
CASP6 P55212 1/20 0.58
MCL1 Q07820 1/20 0.58
PLEC Q15149 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
PGR P06401 2/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
KMT2A Q03164 2/20 0.57
ALDH1A1 P00352 1/20 0.57
TP53 P04637 1/20 0.57
PKM P14618 1/20 0.57
F2 P00734 1/20 0.56
F7 P08709 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15472303 0.96 NR1H4 (0.66) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL18745408 0.91 HPSE (0.57) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL18745403 0.91 KMT2A (0.59) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL15472300 0.91 HPSE (0.57) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL8299942 0.90 NR1H4 (0.67) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL22543145 0.86 NR1H4 (0.78) NR1H4HPSERAB9ANPC1NLRP3
SCHEMBL15472305 0.85 CYP1A2 (0.62) RAB9ANPC1SMN1; SMN2KMT2ATP53
SCHEMBL18745409 0.85 NPC1 (0.67) NR1H4RAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL18745399 0.85 RXFP1 (0.67) RAB9ANPC1NLRP3PGRSMN1; SMN2
SCHEMBL13211973 0.85 NR1H4 (0.68) NR1H4HPSERAB9ANPC1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed