SCHEMBL19860164

SCHEMBL19860164

C/C=C\C1=C(C=O)C2(c3ccccc31)c1ccccc1-c1ccccc12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.36
THRB P10828 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
OPRK1 P41145 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
S100A4 P26447 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21152404 0.88 PDK2 (0.39) PDK2THRBTDP1MEN1KMT2A
SCHEMBL19669965 0.83 PDK2 (0.36) PDK2THRBTDP1MEN1KMT2A
SCHEMBL22435806 0.82 PDK2 (0.35) PDK2THRBTDP1MEN1KMT2A
SCHEMBL21564256 0.81 PDK2 (0.35) PDK2MEN1KMT2AKDM4ELMNA
SCHEMBL21867770 0.80 PDK2 (0.34) PDK2MEN1KMT2AKDM4ELMNA
SCHEMBL21534174 0.78 PDK2 (0.39) PDK2THRBTDP1MEN1KMT2A
SCHEMBL20169416 0.77 PDK2 (0.39) PDK2MEN1KMT2AKDM4ELMNA
SCHEMBL24406310 0.77 PDK2 (0.42) PDK2ESR1ESR2
SCHEMBL21922630 0.77 PDK2 (0.36) PDK2MEN1KMT2AKDM4ELMNA
SCHEMBL20697977 0.77 MEN1 (0.37) PDK2THRBTDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9893299-B2 Heterocyclic compounds MERCK PATENT GMBH (DE) 2018-02-13 US disclosed