SCHEMBL19860193

SCHEMBL19860193

C=CC(=O)Nc1cc(Nc2nc(-c3cn(C)c4ccccc34)c3cc[nH]c3n2)c(OC)cc1N1CCN(C)CC1

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.73
KCNH2 Q12809 3/20 0.60
IGF1R P08069 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17466976 0.91 EGFR (0.70) EGFR
SCHEMBL19860191 0.88 EGFR (0.82) EGFRKCNH2IGF1R
SCHEMBL18921759 0.86 EGFR (0.71) EGFRKCNH2IGF1R
SCHEMBL14718447 0.86 EGFR (0.77) EGFRKCNH2IGF1R
SCHEMBL29974738 0.86 EGFR (0.77) EGFRKCNH2IGF1R
SCHEMBL17467217 0.84 EGFR (1.00) EGFRKCNH2IGF1R
SCHEMBL19239592 0.84 EGFR (0.82) EGFRKCNH2IGF1R
SCHEMBL14663910 0.84 EGFR (0.73) EGFRKCNH2IGF1R
SCHEMBL19860192 0.83 EGFR (0.80) EGFRKCNH2IGF1R
SCHEMBL14719136 0.83 EGFR (1.00) EGFRKCNH2IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890168-B2 2,4-disubstituted 7H-pyrrolo[2,3-d]pyrimidine derivative, preparation method and medicinal use thereof SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2018-02-13 US disclosed
US-9890168-B2 2,4-disubstituted 7H-pyrrolo[2,3-d]pyrimidine derivative, preparation method and medicinal use thereof SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2018-02-13 US disclosed