SCHEMBL1986327

SCHEMBL1986327

C[C@]1(C2CC2)CC2(N=C(N)NC2=O)c2cc(Br)ccc2O1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.49
CTSD P07339 4/20 0.49
APP P05067 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1828909 0.89 BACE1 (0.43) BACE1CTSDAPP
SCHEMBL1821336 0.86 BACE1 (0.65) BACE1CTSD
SCHEMBL1828227 0.81 BACE1 (0.40) BACE1CTSDAPP
SCHEMBL1826421 0.81 BACE1 (0.47) BACE1CTSD
SCHEMBL7960662 0.80 BACE1 (0.44) BACE1CTSDAPP
SCHEMBL7958287 0.79 BACE1 (0.42) BACE1CTSDAPP
SCHEMBL1823413 0.78 BACE1 (0.45) BACE1CTSDAPP
SCHEMBL1832026 0.78 BACE1 (0.45) BACE1CTSD
SCHEMBL7971683 0.78 BACE1 (0.41) BACE1CTSDAPP
SCHEMBL1829335 0.77 BACE1 (0.44) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed