SCHEMBL19866735

SCHEMBL19866735

N#Cc1cnc(N)cc1N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.46
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
LMNA P02545 1/20 0.44
PIK3CA P42336 1/20 0.42
ROCK2 O75116 4/20 0.41
ROCK1 Q13464 4/20 0.41
CDC42BPB Q9Y5S2 4/20 0.41
CDC42BPA Q5VT25 2/20 0.41
CNR2 P34972 2/20 0.39
CNR1 P21554 1/20 0.39
NCF1 P14598 1/20 0.39
CSNK1A1 P48729 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29597546 0.86 PIK3CA (0.57) ALDH1A1MAPTHTTLMNAPIK3CA
SCHEMBL22023334 0.86 PIK3CA (0.57) ALDH1A1MAPTHTTLMNAPIK3CA
SCHEMBL16668734 0.81 FGFR4 (0.45) ARPIK3CAROCK2ROCK1CDC42BPB
SCHEMBL22023340 0.80 PIK3CA (0.42) ARMAPTPIK3CA
SCHEMBL22079818 0.80 PIK3CA (0.41) PIK3CA
SCHEMBL29596603 0.80 PIK3CA (0.41) PIK3CA
SCHEMBL29597799 0.80 PIK3CA (0.42) ARMAPTPIK3CA
SCHEMBL29597907 0.78 LRRK2 (0.38) ARPIK3CAROCK2ROCK1CDC42BPB
SCHEMBL22023291 0.78 LRRK2 (0.38) ARPIK3CAROCK2ROCK1CDC42BPB
SCHEMBL22023223 0.76 ALDH1A1 (0.51) ARALDH1A1MAPTHTTPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018028664-A1 FGFR4 INHIBITOR AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2018-02-15 WO disclosed