SCHEMBL19869905

SCHEMBL19869905

Cc1cc(-c2cn(C)c(=O)c3ccccc23)ccc1C(=O)N1CCN(C)CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.52
BRD9 Q9H8M2 3/20 0.49
BRD7 Q9NPI1 1/20 0.49
CYP2C9 P11712 2/20 0.46
POLB P06746 1/20 0.46
TAF1 P21675 1/20 0.46
CECR2 Q9BXF3 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
TNKS O95271 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19869779 0.86 BRD4 (0.48) BRD4BRD9CYP2C9POLBTAF1
SCHEMBL19869877 0.84 BRD4 (0.69) BRD4CYP2C9POLBTAF1CECR2
SCHEMBL19869921 0.84 BRD4 (0.76) BRD4BRD9TAF1CECR2
SCHEMBL19869828 0.82 BRD4 (0.54) BRD4BRD9CYP2C9POLBTAF1
SCHEMBL19869830 0.82 BRD4 (0.46) BRD4BRD9CYP2C9POLBL3MBTL1
SCHEMBL19869911 0.81 BRD9 (0.56) BRD4BRD9BRD7L3MBTL1
SCHEMBL19869798 0.79 L3MBTL1 (0.46) BRD4BRD9CYP2C9POLBTAF1
SCHEMBL19869908 0.79 BRD9 (0.53) BRD4BRD9BRD7POLBTAF1
SCHEMBL19869918 0.75 BRD4 (0.63) BRD4BRD9TAF1CECR2
SCHEMBL19857641 0.74 BRD4 (0.48) BRD4BRD9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 5/4885BRD9 1/4885BRD7 6/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 6/4885BRD9 1/4885BRD7 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.