SCHEMBL19902113

SCHEMBL19902113

CC1CC2c3sc(NC(=O)Nc4ccc(Cl)cc4)c(C(N)=O)c3CC1N2CC1CCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
TNIK Q9UKE5 1/20 0.42
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
TP53 P04637 1/20 0.37
XBP1 P17861 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17018790 0.84 KCNH2 (0.54) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL17018788 0.82 KCNH2 (0.53) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL18902174 0.79 KCNH2 (0.49) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL17018791 0.76 KCNH2 (0.58) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL16961226 0.75 KCNH2 (0.72) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL19807401 0.74 KCNH2 (0.71) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL18012600 0.74 KCNH2 (0.71) KCNH2CYP3A4CYP2C9CYP2C19TNIK
Hydrochloric Acid SCHEMBL17006410 0.74 KCNH2 (0.73) KCNH2CYP3A4CYP2C9CYP2C19TNIK
SCHEMBL19807539 0.74 KCNH2 (0.56) KCNH2CYP3A4CYP2C9CYP2C19TNIK
Hydrochloric Acid SCHEMBL17969205 0.73 KCNH2 (0.71) KCNH2CYP3A4CYP2C9CYP2C19TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902738-B2 Compounds and methods for preventing, treating and/or protecting against sensory hair cell death UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2018-02-27 US disclosed